Екип

Координатор на консорциума

Членове на научния колектив

 

д-р Георги Цветанов Момеков, д.м.

Организация, контакти:

Медицински Университет София
Фармацевтичен факултет
Катедра „Фармакология, Фармакотерапия и Токсикология”

София 1000, ул. „Дунав” №2
тел: (02) 9236509

email: gmomekov@cetrh.org

Членства в научни организации:
  • Българско научно дружество по фармация, Член на управителния съвет
  • Национално научно дружество по токсикология
  • Национално научно дружество по фармакология
  • Български фармацевтичен съюз
Научни награди: “Signum Laudis ad Scientiae Meritis”, присъдена от Съвет по медицинска наука, МУ-София
Основни публикации
  1. Momekov, G., Ferdinandov,D., Zheleva-Dimitrova,D., Nedialkov,P., Girreser, U., Kitanov,G. Cytotoxic effects of
    hyperatomarin, a prenylated phloroglucinol from Hypericum annulatum Moris subsp. annulatum, in a panel of
    malignant cell lines (2008) Phytomedicine (In press)
  2. Karaivanova, M., Kostovski, A., Momekov, G. Angiogenesis and approaches to designing antiangiogenic drugs
    (2008) Pharmacia (Sofia) (In press)
  3. Momekov, G., Ferdinandov, D., Konstantinov, S., Arpadjan, S., Tsekova, D., Gencheva, G., Bontchev, P.R.,
    Karaivanova, M. In vitro evaluation of a stable monomeric gold(II) complex with hematoporphyrin IX:
    Cytotoxicity against tumor and kidney cells, cellular accumulation and induction of apoptosis (2008) Metal Based
    Drugs, 2008 Article ID 367471, 8 pages doi:10.1155/2008/367471
  4. Bakalova, A., Varbanov, H., Momekov, G. Palladium(II) complexes with 5-methyl-5-(4-pyridyl)-2,4-
    imidazolidinedione. Synthesis, thermogravimetric and cytotoxic investigation. (2008) Journal of Thermal Analysis
    and Calorimetry (In press).
  5. Kostova, I., Trendafilova, N., Momekov, G. Theoretical, spectral characterization and antineoplastic activity of
    new lanthanide complexes (2008) Journal of Trace Elements in Medicine and Biology (In Press)
  6. Stanchev, S., Momekov, G., Jensen, F., Manolov.I. Synthesis, computational study and cytotoxic activity of new 4-
    hydroxycoumarin derivatives. (2008) European Journal of Medicinal Chemistry, 43 (4) pp. 694-706.
  7. Kostova, I., Momekov, G. New cerium(III) complexes of coumarins – Synthesis, characterization and cytotoxicity
    evaluation (2008) European Journal of Medicinal Chemistry, 43 (1) pp. 178-188
  8. Ivanova, J.B., Momekov, G.Ts., Kalcheva, V.B., Petrov, O.I. Synthesis of chalcones condensed with an 1,3-azole
    ring using a SOCl2/EtOH catalytic system.(2008) Comptes Rendus de’l Academie Bulgare des Sciences 61 (1) pp.
    41-48.
  9. Momekov, G., Todorov, P., Naydenova, E., Kostovski, A., Troev, K. Cytotoxic activity of new α-aminophosphonic
    acids against human malignant cell lines (2007) Pharmacia (Sofia) 54 (3-4) pp. 9-11.
  10. Kostova, I., Kiefer, W., Momekov, G. Cytotoxic activity of Gd(III) and Dy(III) – complexes
    (2007) Archive die Pharmazie (Weinheim) 340 (12) pp.642-9.
  11. Nikolov, S., Momekov, G., Kitanov, G., Ionkova, I., Krasteva, I., Toshkova, R., Konstantinov, S., Nedialkov, P.,
    Karaivanova, M. Exploitation of the Bulgarian Flora’s biodiversity as a source of immunomodulatory and/or
    antineoplastic agents: Current challenges and perspectives. (2007) Biotechnology & Biotechnological Equipment
    21 (4) pp. 471-477.
  12. Momekova, D., Momekov, G., Rangelov, S., Lambov, N. In vitro biocompatibility study of free and liposomalygrafted
    copolymers bearing short blocks of aliphatic lipid-mimetic units – cytotoxicity and hemolytic activity.
    (2007) Journal of Drug Delivery Science and Technology 17(6) pp.393-397.
  13. Ivanova, Y.B., Gerova, M.S., Momekov, G.Ts., Petrov, O.I. Synthetic chalcones of 2(3H)-benzothiazolone with
    potential cytotoxic activity. (2007) Comptes Rendus de’l Academie Bulgare des Sciences 60 (6) pp. 641-644.
  14. Krasteva, I., Platikanov, S., Momekov, G., Konstantinov, S., Nikolov, S. Phytochemical analysis and in vitro
    cytotoxic activity of volatiles from Astragalus corniculatus. (2007) Natural Product Research (In press).ю
  15. Naydenova, E., Todorov, P.T., Topashka-Ancheva, M., Momekov, G. Ts., Yordanova, T.Z., Konstantinov, S.M.,
    Troev, K.D. Novel N-(phosphonomethyl) glycine derivatives. Design, characterization and biological activity.
    (2008) European Journal of Medicinal Chemistry 43, pp.1199-1205.
  16. Bakalova, A., Varbanov, H., Buyukliev, R., Momekov, G., Ferdinandov, D., Konstantinov, S., Ivanov, D.
    Synthesis, characterization and biological activity of Pt(II) and Pt(IV) complexes with 5-methyl-5(4-pyridyl)-2,4-
    imidazolidenedione. (2008) European Journal of Medicinal Chemistry, 43, pp. 958-965.
  17. Momekov, G., Krasteva, I., Platikanov, S., Nikolov, S., Konstantinov, S. Cytotoxic activity of volatiles from four
    Astragalus species. (2007) Comptes Rendus de’l Academie Bulgare des Sciences 60 (9) pp. 1023-1026.
  18. Gencheva, G., Tsekova, D., Gochev, G., Momekov, G., Tyuliev, G., Skumryev, V., Karaivanova, M., Bontchev,
    P.R. Synthesis, structural characterization and cytotoxic activity of novel paramagnetic platinum hematoporphyrin
    complexes – potent antitumour agents (2007) Metal-Based Drugs 2007 Article ID 67376, 13 Pages, doi
    10.1155/2007/67376
  19. Ionkova, I., Antonova, I., Momekov, G., Fuss, E. Cytotoxic activity of extracts from Bulgarian Linum species.
    (2007) Pharmacognosy Magazine, 3 (11) pp. 192-195.
  20. Ivanova, Y., Momekov, G., Petrov, O., Karaivanova, M., Kalcheva, V. Cytotoxic Mannich bases of 6-(3-aryl-2-
    propenoyl)-2(3H)-benzaxolones. (2007) European Journal of Medicinal Chemistry, 42 (11-12) pp.1382-1387.
  21. Kostova, I., Momekov, G. Synthesis, characterization and cytotoxicity determination of new cerium(III),
    lanthanum(III) and neodymium(III) complex compounds. (2007) Applied Organometallic Chemistry, 21(4), pp.
    226-233.
  22. Kostova, I. Trendafilova, N., Cinta Pinzaru, S., Kiefer, W., Momekov, G.
    Spectroscopic evidence of La(III) complex of coumarin-3-carboxylic acid with cytotoxic activity. (2007) Journal
    of Optoelectronics and Advanced Materials, 9(3), pp. 532-539.
  23. Kostova, I., Momekov, G., Stancheva, P. New samarium(III), gadolinium(III) and dysprosium(III) complexes of
    coumarin-3-carboxylic acid as cytotoxic agents. (2007) Metal-Based Drugs 2007, Article ID 15925, 8 pages;
    doi:10.1155/2007/15925
  24. Momekov, G., Konstantinov, S., Bakalova, A., Topashka-Ancheva, M., Arpajan, S. Karaivanova, M. Cellular
    pharmacology, antineoplastic activity and low in vivo toxicity of a carboxylato-bridged platinum(II) complex bisacetatodiammine-
    bis-μ-acetato diplatinum(II) dihydrate.(2007) Medicinal Chemistry, 3 (2), pp. 157-165.
  25. Momekov, G., Momekova, D. Recent developments in antitumour platinum coordination compounds. (2006)
    Expert Opinion on Therapeutic Patents, 16 (10), pp. 1383-1403.
  26. Momekov, G., Deligeorgiev, T., Vasilev, A., Peneva, K., Konstantinov, S., Karaivanova, M.
    Evaluation of the cytotoxic and pro-apoptotic activities of Eu(III) complexes with appended DNA intercalators in a
    panel of human malignant cell lines (2006) Medicinal Chemistry, 2 (5), pp. 439-445.
  27. Momekov, G., Ferdinandov,D., Bakalova,A., Zaharieva,M., Konstantinov, S., Karaivanova,M.
    In vitro toxicological evaluation of a dinuclear platinum(II) complex with acetate ligands (2006) Archives of
    Toxicology, 80 (9), pp. 555-560.
  28. Kostova, I., Momekov, G. New zirconium (IV) complexes of coumarins with cytotoxic activity (2006) European
    Journal of Medicinal Chemistry, 41 (6), pp. 717-726.
  29. Momekov, G., Nedialkov, P.T., Kitanov, G.M., Zh. Zheleva-Dimitrova, D., Tzanova, T., Girreser, U., Karaivanova,
    M. Cytoprotective effects of 5 benzophenones and a xanthone from Hypericum annulatum in models of epirubicininduced
    cytotoxicity: SAR-analysis and mechanistic investigations (2006) Medicinal Chemistry, 2 (4), pp. 377-384.
  30. Vasilev, N., Elfahmi, Bos, R., Kayser, O., Momekov, G., Konstantinov, S., Ionkova, I.
    Production of justicidin B, a cytotoxic arylnaphthalene lignan from genetically transformed root cultures of Linum
    leoni (2006) Journal of Natural Products, 69 (7), pp. 1014-1017.
  31. Manolov, I., Machulla, H.-J., Momekov, G. Synthesis, physicochemical characterization and preliminary
    pharmacological in vitro evaluation of two novel cytotoxic benzophenone-linked 3,3-dimethyltriazenes (2006)
    Pharmazie, 61 (6), pp. 511-516.
  32. Kostova, I., Momekov, G., Tzanova, T., Karaivanova, M. Synthesis, characterization, and cytotoxic activity of new
    lanthanum(III) complexes of bis-coumarins (2006) Bioinorganic Chemistry and Applications, 2006, art. no. 25651,
  33. Todorov, P., Naydenova, E., Momekov, G., Troev, K. Antitumor activity of new alpha-aminophosphonic acids and
    oligopeptides. (2006) Proceedings of the 29-th European Peptide Symposium, Gdansk, Poland, September 3-8
    2006.
  34. Momekov, G., Bakalova, A., Konstantinov, S., Todorov, D., Karaivanova, M. Comparative assessment of the
    cytotoxic effects of carboxylato-bridged dinuclear platinum (II) complexes against human tumor cell lines (2005)
    Neoplasma, 52 (6), pp. 469-475.
  35. Kostova, I., Manolov, I., Momekov, G., Tzanova, T., Konstantinov, S., Karaivanova, M. Cytotoxic activity of new
    cerium (III) complexes of bis-coumarins (2005) European Journal of Medicinal Chemistry, 40 (12), pp. 1246-1254.
  36. Vasilev, N., Momekov,G., Zaharieva, M.,Konstantinov, S., Bremner, P.,Heinrich, M., Ionkova, I. Cytotoxic
    activity of a podophyllotoxin-like lignan from Linum tauricum Willd (2005) Neoplasma, 52 (5), pp. 425-429.
  37. Momekov, G., Bakalova, A., Karaivanova, M. Novel approaches towards development of non-classical platinumbased
    antineoplastic agents: Design of platinum complexes characterized by an alternative DNA-binding pattern
    and/or tumor-targeted cytotoxicity (2005) Current Medicinal Chemistry, 12 (19), pp. 2177-2191.
  38. Zaharieva, M., Petkov,N., Pilicheva,B., Yosifov,D., Momekov,G., Konstantinov,S., Berger,M.
    Evaluation of the combined effects of erucylphospho-N,N,N,-trimethylpropylammonium (ERPC3), gleevec and
    bendamustine on normal and malignantly transformed haemopoietic cells (2005) Pharmacia (Sofia), 52 (1-2), pp.
    90-98.
  39. Bakalova, A., Buyukliev, R., Momekov, G., Ivanov, D., Todorov, D., Konstantinov, S., Karaivanova, M. Synthesis,
    physicochemical and in vitro pharmacological investigation of new platinum (II) complexes with some
    cycloalkanespiro-5`-hydantoins. (2005) European Journal of Medicinal Chemistry, 40 (6), pp. 590-596.
  40. Kostova, I., Momekov, G., Zaharieva, M., Karaivanova, M. Cytotoxic activity of new lanthanum (III) complexes of
    bis-coumarins. (2005) European Journal of Medicinal Chemistry, 40 (6), pp. 542-551.
  41. Kostova, I., Kostova, R., Momekov, G., Trendafilova, N., Karaivanova, M. Antineoplastic activity of new
    lanthanide (cerium, lanthanum and neodymium) complex compounds. (2005) Journal of Trace Elements in
    Medicine and Biology, 18 (3), pp. 219-226.
  42. Kostova, I., Trendafilova, N., Momekov, G. Theoretical and spectroscopic evidence for coordination ability of 3,3’-
    benzylidenedi-4-hydroxycoumarin. New neodymium (III) complex and its cytotoxic effect. (2005) Journal of
    Inorganic Biochemistry, 99 (2), pp. 477-487.
  43. Kostova, I., Manolov, I., Momekov, G. Cytotoxic activity of new neodymium (III) complexes of biscoumarins. (2004) European Journal of Medicinal Chemistry, 39 (9), pp. 765-775.